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Intermediates

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Intermediates

API name Intermediates CAS number
Sapropterin dihydrochloride sapropterin dihydrochloride 69056-38-8
l-erythro biopterin  22150-76-1
PtO2 1314-15-4
Vumerity(Diroximel fumarate) Diroximel fumarate 1577222-14-0 
Monomethyl  fumarate 2756-87-8
N-(2-hydroxyethyl) succinimide 18190-44-8
1-Ethyl-3-(3-dimethylaminopropyl)carbodoomid hydrochloride 25952-53-8
DBU   6674-22-2
Roxadustat Roxadustat 808118-40-3
Methyl 4-hydroxy-1-methyl-7-phenoxyisoquinoline-3-carboxylate 1421312-34-6
Glycine 56-40-6
DBU 6674-22-2
 Ruxolitinib Phosphate (R)-3-Cyclopentyl-3-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl)propanenitrile  1146629-84-6
 4-chloro-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidine 16372-08-0
Palladium-tetrakis(triphenylphosphine) Pd(PPh3)4 14221-01-3
Favipiravir  3,6-Dichloropyrazine-2-carbonitrile 356783-16-9
Potassium fluoride dihydrate 13455-21-5
TBAB 1643-19-2
Cladribine  
2-chloro-6-amino-9-(3,5-di-O-p-toluoyl-2-deoxy-β-D-erythropentofuranosyl) purine
39031-33-9
1-chloro-3,5-di-toluoyl-2-deoxy-D-ribose 3601-89-6
2-Chlorophenthiazine 1839-18-5
Fingolimode N-[1,1-Bis[(acetyloxy)methyl]-3-(4-octylphenyl)propyl]acetamide 162358-09-0
Ozanimod Hcl (S)-tert-butyl (2-((tert-butyldimethylsilyl)oxy)ethyl)(4-(N-hydroxycarbamimidoyl)-2,3-dihydro-1H-inden-1-yl)carbamate 1306763-62-1
 
3-Cyano-4-isopropoxy-benzoic acid
258273-31-3
1-Hydroxy benzotriazole monohydrate 123333-53-9
N3-dimethylpropane-1,3-diamine hydrochloride 25952-53-8
Siponimod fumaric acid   
4-{1-[(E)-4-cyclohexyl-3-trifluoromethyl-benzyloxyimino]-ethyl}-2-ethyl-benzyldehyde
1230487-01-0
 
azetidine-3-carboxylic acid
36476-78-5
ETHYL CYANOACETATE 105-56-6
Enzalutamide 4-Isothiocyanato-2-(trifluoromethyl)benzonitrile 143782-23-4
2-(3-fluoro-4-(methylcarbamoyl)phenylamino)-2-methylpropanoate 1332524-01-2
Netupitant 6-(4-Methylpiperazin-1-yl)-4-(2-methylphenyl)nicotinamide 342417-01-0
2-(3,5-bis(trifluoroMethyl)phenyl)-2-Methyl propanoic acid 289686-70-0
Indacaterol 5,6-Diethyl-2,3-dihydro-1H-inden-2-amine hydrochloride 312753-53-0
Delafloxacin 3,5-Difluoropyridine-2,6-diamine 247069-27-8
Bilastine 2-methyl-2-(4-(2-(tosyloxy)ethyl)phenyl)propanoate 1181267-30-0
4-(1-(2-ethoxyethyl)-1H-benzo[d]iMidazol-2-yl)piperidine-1-carboxylate 1181267-36-6
Alcaftadine 1-Phenethylimidazole 49823-14-5
1-(Ethoxycarbonyl)piperidine-4-carboxylic acid 118133-15-6
11-(1-Methylpiperidin-4-ylidene)-6,11-dihydro-5H-benzo[d]iMidazo[1,2-a]azepine 147083-36-1
Azelastine hydrochloride 4-hydrazineyl-1-methylazepane hydrogen chloride  
Formoterol N-Benzyl-1-(4-methoxyphenyl)propan-2-amine hydrochloride 1049695-95-5
2-Bromo-4'-Benzyloxy-3'-nitroacetophenone 43229-01-2
Olaparib 2-Fluoro-5-[(3-oxo-1(3H)-isobenzofuranylidene)methyl]-benzonitrile 763114-25-6
2-Fluoro-5-formylbenzonitrile  218301-22-5 
5-[(3,4-Dihydro-4-oxo-1-phthalazinyl)methyl]-2-fluoro-Benzoic acid 763114-26-7
Crizotinib 4-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]-, 1,1-dimethylethyl ester 877399-74-1
(S)-1-(2,6-Dichloro-3-fluorophenyl)ethanol 877397-65-4
2-Nitro-3-hydroxypyridine 15128-82-2
5-bromo-3-[(1R)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]pyridin-2-amine 877399-00-3
Palbociclib  3-aminophthalic acid hcl dihydrate 6946-22-1
6-broMo-2-chloro-8-cyclopentyl-5-Methylpyrido[2,3-d]pyriMidin-7(8H)-one 1016636-76-2
Rivaroxaban 4-(4-Aminophenyl)morpholin-3-one 438056-69-0
5-Chloro-2-thiophenecarboxylic acid 24065-33-6
5-Chlorothiophene-2-carbonyl chloride 42518-98-9
(S)-(+)-Glycidyl phthalimide 161596-47-0
(S)-4-(4-(5-(Aminomethyl)-2-oxooxazolidin-3-yl)phenyl)morpholin-3-one HCl 898543-06-1
2-[[(5S)-2-Oxo-3-[4-(3-oxo-4-morpholinyl)phenyl]-5-oxazolidinyl]methyl]-1H-isoindole-1,3(2H)-dione 446292-08-6
Rivaroxaban 366789-02-8
Isavuconazole 2-Bromo-4'-cyanoacetophenone 20099-89-2
Lorcaserin hydrochloride 1-[[2-(4-Chlorophenyl)ethyl]aMino]-2-chloropropane 953789-37-2
Lorcaserin hydrochloride 846589-98-8
Lorcaserin hydrochloride hemihydrate 856681-05-5
Bortezomib (aR,3aS,4S,6S,7aR)-Hexahydro-3a,8,8-trimethyl-alpha-(2-methylpropyl)-4,6-methano-1,3,2-benzodioxaborole-2-methanamine 2,2,2-trifluoroacetate 179324-87-9
(S)-3-Phenyl-2-[(pyrazin-2-ylcarbonyl)amino] propanoic acid 114457-94-2
Isobutaneboronic acid 84110-40-7
8-Bromooctanoic Ethylester 29823-21-0
Bortezomib 179324-69-7
APAXIBAN Ethyl1-(4-Methoxyphenyl)-7-oxo-6-[4-(2-oxopiperidin-1-yl)phenyl]-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylic acid  ester 503614-91-3
Oxcarbazepine 10-Methoxyiminostilbene 4698-11-7
Tazarotene 6-Acetyl-4,4-dimethylthio-chroman 18579-23-1
6-Ethynyl-4,4-dimethylthiochroman 118292-06-1
Tazarotene 118292-40-3
Tapentadol Hydrochloride 3'-Hydroxypropiophenone 13103-80-5
3-Bromoanisole 2398-37-0
3'-methoxypropiophenone 37951-49-8
Paliperidone 3-(2-Chloroethyl)-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one 130049-82-0
Paliperidone 144598-75-4
Tofacitinib N-Methyl-N-((3R,4R)-4-Methylpiperidin-3-yl)-7H-pyrrolo[2,3-d]pyriMidin-4-aMine   477600-74-1
Carfilzomib (2s)-2-amino-4-methyl-1-((2r)-2-methyloxiranyl)-1-pentanone trifluoroacetate 247068-85-5
(alphaS)-alpha-[(4-Morpholinylacetyl)aMino]benzenebutanoyl-L-leucyl-L-phenylalanine 868540-16-3
Etoricoxib 2-(4-Methanesulfonyl-phenyl)-1-(6-methyl-pyridin-3-yl)-ethanone 221615-75-4
2-Chloro-1,3-bis(dimentylamino) trimethinium hexafluorophosphate 249561-98-6
Conivaptan hydrochloride 2-Methyl-1,4,5,6-tetrahydroimidazo[4,5-d][1] benzazepine 318237-73-9
Dabigatran etexilatemesilate N-[2-[4-[N-(Hexyloxycarbonyl)amidino] phenylaminomethyl]-1-methyl-1H-benzimidazol-5-ylcarbonyl]-N-(2-pyridyl)-beta-alanine ethyl ester 211915-06-9
N-[[2-[[[4-[[[(Hexyloxy)carbonyl] amino]iminomethyl]phenyl]amino]methyl]-1-methyl-1H-benzimidazol-5-yl]carbonyl]-N-2-pyridinyl-beta-alanine ethyl ester monomethanesulfonat 872728-81-9
3-[(3-Amino-4-Methylamino-Benzoyl)-Pyridin-2-Yl-Amino]-Propionic Acid Ethyl Ester 212322-56-0
N-(4-Cyano-Phenyl)-Glycine 42288-26-6
3-[[[2-[[(4-Cyanophenyl)amino]methyl]-1-methyl-1H-benzimidazol-5-yl]carbonyl]pyridin-2-ylamino]propionic acid ethyl ester 211915-84-3
3-[[2-[[(4-carbamimidoylphenyl) amino]methyl]-1-methyl-benzoimidazole-5-carbonyl]-pyridin-2-yl-amino]propanoic acid 211914-51-1
Argatroban  3-Methyl-8-quinolinesulphonyl chloride 74863-82-4
Pimavanserin 4-(2-methylpropoxy)-benzenemethanamine hydrochloride 54799-03-0
N-(4-fluorobenzyl)-1-methylpiperidin-4-amine 359878-47-0 
Nilotinib 4-Methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]benzoic acid 641569-94-0
1-(3-Pyridyl)-3-(dimethylamino)-2-propen-1-one  55314-16-4
3-(4-Methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)
aniline 
641571-11-1
GS 7340 GS 7340 fumarate
N-[(S)-[[(1R)-2-(6-Amino-9H-purin-9-yl)-1-methylethoxy]methyl] phenoxyphosphinyl]-L-llanine 1-methylethyl ester (2E)-2-butenedioate (1:1)
379270-38-9
Teneligliptin (2S)-4-Oxo-2-(3-thiazolidinylcarbonyl)-1-pyrrolidinecarboxylic acid tert-butyl ester 401564-36-1
1-(3-Methyl-1-phenyl-5-pyrazolyl)piperazine 401566-79-8
Teneligliptin 760937-92-6
Moxonidine  Ethanone 75438-54-9
 5-Amino-4,6-dichloro-2-methylpyrimidine 39906-04-2
Oseltamivir Phosphate Oseltamivir Phosphate 204255-11-8
Remdesivir  ACS9087-10 1191578-98-7
ACS9087-13 1191237-69-0
Peramivir Methyl (1S,4R)-4-[(tert-butoxycarbonyl)amino]cyclopent-2-ene-1-carboxylate 229613-93-8
(1S,2S,3S,4R)-methyl3-((R)-1-amino-2-ethylbutyl)-4-(tert-butoxycarbonylamino)-2-hydroxycyclopentanecarboxylat 316173-29-2
Obeticholic 3α-hydroxy-6-ethyliden-7-keto-5β-cholan-24-oate 863239-59-2
(E)-3-hydroxy-6-ethylidene-7-keto-5-cholan-24-oic acid 1516887-33-4
1osv 459789-99-2
Bazedoxifene Acetate Bazedoxifene intermediate I 198479-63-9
1-[2-(4-chloromethyl-phenoxy)-ethyl]-azepane hydrochloride 223251-25-0
Bazedoxifene intermediate I 198480-21-6
Baloxavir 1H-[1,4]Oxazino[3,4-c]pyrido[2,1-f][1,2,4]triazine-6,8-dione, 3,4,12,12a-tetrahydro-7-(phenylmethoxy)- 1370250-39-7
1H-[1,4]Oxazino[3,4-c]pyrido[2,1-f][1,2,4]triazine-6,8-dione, 3,4,12,12a-tetrahydro-7-(phenylmethoxy)-, (12aR)- 1985607-70-2
Dibenzo[b,e]thiepin-11-ol, 7,8-difluoro-6,11-dihydro- 1985607-83-7
Dibenzo[b,e]thiepin-11(6H)-one, 7,8-difluoro- 2136287-66-4
Bictegravir (1R,3S)-3-Aminocyclopentanolhydrochloride;(1R,3S)-3-aminocyclopentanol hydrochloride 1279032-31-3
2,3-DIHYDROXY-3-(5-METHYL-1H-BENZOIMIDAZOL-2-YL)-PROPIONIC ACID 214759-21-4
Velpatasvir GS 5816 1377049-84-7
 
tert-butyl(2S,4S)-2-(5-(2-((2S,5S)-1-((methoxycarbonyl)-L-valyl)-5-methylpyrrolidin-2-yl)-1,11-dihydroisochromeno[4',3':6,7]naphtho[1,2-d]imidazol-9-yl)-1H-imidazol-2-yl)-4-(methoxymethyl)pyrrolidine-1-carboxylate;
1378391-45-7
Sofosbuvir Cytidine, N-benzoyl-2'-deoxy-2'-fluoro-2'-methyl-, 3',5'-dibenzoate, (2'R)-  817204-32-3
2'-deoxy-2'-fluoro-2'-C-Methyluridine  863329-66-2
Ledipasvir Ledipasvir Impurity 8 1256387-74-2

(S)-5-BOC-5-AZASPIRO[2.4]HEPTANE-6-CARBOXYLIC ACID
1129634-44-1
ledipasvir interMediate 1441670-89-8

Ledipasvir
1256388-51-8

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